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找到约 32 条 “OX Receptor” 相关结果（用时 0.142 秒）

目录号	产品名称	中文名称	靶点
M21445	Recombinant Human OLR1/LOX1 (Mammalian, C-6His)	重组人OLR1/LOX1蛋白 (Mammalian, C-6His)	Recombinant Proteins
	Oxidized Low-Density Lipoprotein Receptor 1; LOX-1
	Oxidized low-density lipoprotein receptor 1 (Ox-LDL receptor 1 or OLR1), also known as LOX1, is a receptor protein that belongs to the C-type lectin superfamily. LOX1 may play an important role in the progression of vulnerable carotid plaque and might regulate vulnerable plaque formation in cooperation with MMPs and TIMP-2.
M29995	OT-R antagonist 1	OT-R antagonist 1	Oxytocin Receptor
	Oxytocin receptor antagonist 1
	OT-R antagonist 1是一种新型有效的选择性非肽类OT-R拮抗剂, 抑制催产素诱发的细胞内Ca2+活动（IC50=8nM）。
M2088	Ciproxifan maleate	Ciproxifan maleate	Histamine Receptor
	FUB 359 maleate
	Ciproxifan（CPX）是一种高效的，选择性的histamin H3-receptor拮抗剂，IC50为9.2 nM，作用于其他受体亚型具有低亲和力。
M2105	Azilsartan medoxomil	阿齐沙坦酯	Angiotensin Receptor
	TAK-491
	Azilsartan Medoxomil是一种有效的angiotensin II type 1 (AT1) receptor（血管紧张素II 1型受体）拮抗剂，抑制RAAS比作用于AT2选择性高10，000倍以上，用于研究高血压。
M2280	Tamoxifen Citrate (ICI 46474)	柠檬酸三苯氧胺；柠檬酸它莫西芬；柠檬酸他莫昔芬	Estrogen Receptor
	ICI 46474; Istubal; Nolvadex
	Tamoxifen Citrate是一种雌激素受体（Estrogen Receptor）拮抗剂，与雌激素竞争性结合。
M2507	Chenodeoxycholic acid	鹅去氧胆酸	Farnesoid X Receptor
	CDCA; Chenodiol
	Chenodeoxycholic Acid是一种天然存在的人体胆汁酸，也是一种法尼类X受体（Farnesoid X Receptor）的激动剂。可用于脑腱黄瘤病(CTX)的相关研究。
M2522	Ciproxifan	Ciproxifan	Histamine Receptor
	FUB-359
	Ciproxifan（CPX）是一种高效的，选择性的histamin H3-receptor拮抗剂，IC50为9.2 nM，作用于其他受体亚型具有低亲和力。
M2842	Methoxamine hydrochloride	凡索昔；美迷克新命；盐酸甲氧胺；盐酸甲氧明	Adrenergic Receptor
	Vasoxine HCl
	Methoxamine是一种α1-肾上腺素能受体（α1-adrenergic receptor）激动剂，它能诱导皮肤和脾脏血管收缩。
M3324	SB408124	SB408124	OX Receptor
	SB408124是一种非肽类OX1 receptor拮抗剂，作用于全细胞和膜，K_i分别为57 nM和27 nM，比作用于OX2受体选择性高50倍。
M3413	Phenoxybenzamine hydrochloride	盐酸酚苄明	Adrenergic Receptor
	Phenoxybenzamine HCl（盐酸酚苄明）是一种非选择性的，不可逆α肾上腺素能受体（Adrenergic Receptor）拮抗剂，IC50为550 nM。
M1565	Quetiapine sulfoxide	喹硫平硫氧化物/喹硫平亚砜	5-HT Receptor
	Quetiapine sulfoxide; Quetiapine S-oxide
	Quetiapine sulfoxide是一种 5-HT 受体激动剂，对人 5-HT1A 的 pEC50 值为 4.77。Quetiapine hemifumarate 是多巴胺受体 (dopamine receptor) 拮抗剂，对人 D2 的 pIC50 值为 6.33。
M4887	Pardoprunox Hydrochloride	盐酸帕多芦诺	5-HT Receptor
	SLV-308
	Pardoprunox hydrochloride (DU-126891, SME-308)是一种有效的部分 dopamine D2 receptor 的激动剂，对应的pEC50值为8.0，也是诱导 [35S]GTPγS binding 的部分激动剂，对应的pEC50值为9.2，和 serotonin 5-HT1A receptor 的激动剂，pEC50值为6.3。
M6720	Etifoxine hydrochloride	盐酸艾替伏辛	GABA Receptor
	HOE 36-801
	Etifoxine hydrochloride is a ligand of the translocator protein (TSPO); also GABA _A receptor potentiator.
M6833	IPSU	IPSU	OX Receptor
	IPSU is a oX ₂ receptor antagonist; orally bioavailable.
M7174	PTAC oxalate	PTAC oxalate	Others
	PTAC oxalate is a muscarinic receptor ligand; exhibits partial agonist and antagonist activity at different subtypes.
M7213	Roxindole hydrochloride	Roxindole hydrochloride	Others
	Roxindole hydrochloride is a dopamine D ₂ autoreceptor agonist. Also has affinity for D ₃, D ₄, 5-HT _1A receptors and the 5-HT transporter.
M7353	Tamoxifen	他莫昔芬	Estrogen Receptor
	ICI47699; Z-Tamoxifen; trans-Tamoxifen
	Tamoxifen是一种选择性雌激素受体调节剂 (Selective estrogen receptor modulators，SERM)，可阻断乳腺细胞中的雌激素作用。Tamoxifen 也是一种有效的 Hsp90 激活剂，可增强 Hsp90 分子伴侣 ATPase 的活性。Tamoxifen 还可以有效抑制传染性 EBOV Zaire 和 Marburg (MARV)，IC50 分别为 0.1 µM 和 1.8 µM。
M7439	U 46619	U 46619	Others
	U 46619 is a potent, stable thromboxane A ₂ (TP) receptor agonist.
M7722	Ciproxifan hydrochloride	环丙基[4-[3-(1H-咪唑-5-基)丙氧基]苯基]甲酮盐酸盐	Others
	Ciproxifan（CPX） belongs to a novel chemical series of histamine H₃-receptor antagonists.
M7769	Daltroban	达尔卓潘	Others
	Selective thromboxane A₂ receptor antagonist.
M7855	ICI 192605	ICI 192605	Others
	ICI 192605 is a potent thromboxane A2 receptor antagonist.
M7946	Naloxone methiodide	Naloxone methiodide	Others
	Quaternary salt of naloxone that, like the parent compound, is a nonselective antagonist at opioid receptors.
M8048	Nafoxidine hydrochloride	盐酸萘福昔定	Others
	Nafoxidine is a potent estrogen receptor antagonist that exhibits anti-proliferative properties.
M8139	Ridaifen-B	Ridaifen-B	Others
	Ridaifen-B (RID-B) is a novel tamoxifen (TAM) analog that significantly augments apoptosis-inducing effect of TAM in estrogen receptor (ER)-negatives cells.
M8150	SB-668875	SB-668875	Others
	SB-668875 is a novel, selective peptide agonist at OX2 orexin receptors.
M8234	Loxiglumide	氯谷胺	Others
	CR-1505
	Loxiglumide is a small-molecule antagonist of the cholecystokinin receptor CCKA.
M8366	DDN	DDN	Others
	DDN (5,8-Diacetyloxy-2,3-dichloro-1,4-naphthoquinone) is a selective insulin receptor (IR) activator that binds directly to the receptor kinase domain and induces the Akt and ERK phosphorylations.
M8416	Darglitazone sodium salt	Darglitazone sodium salt	Others
	Darglitazone is a highly potent and selective PPAR-γ (peroxisome proliferator-activated receptor-γ) agonist.
M8482	Nonyloxytryptamine oxalate	Nonyloxytryptamine oxalate	Others
	Nonyloxytryptamine (5-nonyloxytryptamine) is a potent and selective 5-HT1B receptor agonist.
M9674	MRS-3777 hemioxalate	MRS-3777 hemioxalate	Adenosine Receptor
	MRS-3777 hemioxalate是一种选择性的腺苷A3受体（adenosine A3 receptor）拮抗剂。
M10348	27-Hydroxycholesterol	27-羟基胆固醇	Estrogen Receptor
	27-Hydroxycholesterol是一种选择性的雌激素受体 (estrogen receptor) 调节剂，它也是一种肝脏X受体 (liver X receptor) 的激动剂。
M11259	Cefminox sodium	头孢米诺钠	Antibiotic
	Meicelin, MT-141
	Cefminox sodium (MT-141) 是一种半合成的头霉素，具有广谱的抗菌活性。Cefminox sodium (MT-141) 为前列环素受体 (prostacyclin receptor) 和 PPARγ 的双重激动剂，能够上调 cAMP 的产生和 PTEN 的表达，抑制 Akt/mTOR 信号通路。Cefminox sodium (MT-141) 可抑制肺动脉高压。

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